Document Type

Article

Keywords

Carbohydrates, Glycosylation, Leaving group, Oligosaccharides, Orthogonal strategy, Selective activation

Abstract

The O-allylphenyl (AP) anomeric moiety was investigated as a new leaving group that can be activated for chemical glycosylation under a variety of conditions, through both direct and remote pathways. Differentiation between the two activation pathways was achieved in a mechanistic study. The orthogonal-type activation of the AP moiety along with common thioglycosides allows for the execution of efficient oligosaccharide assembly. © 2012 Premathilake and Demchenko.

Publication Date

4-26-2012

Publication Title

Beilstein Journal of Organic Chemistry

E-ISSN

18605397

Volume

8

First Page

597

Last Page

605

Rights

CC BY

DOI

10.3762/bjoc.8.66

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